Bioorganic and Medicinal Chemistry Letters Journal

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Dimers of isatin derived -methylene--butyrolactone as potent anti-cancer agents.. 65:128713-128713. 2022
New -lactam - Tetramic acid hybrids show promising antibacterial activities.. 28:3105-3112. 2018
Part 2. Notch-sparing -secretase inhibitors: The study of novel -amino naphthyl alcohols.. 26:2133-2137. 2016
Part 1: Notch-sparing -secretase inhibitors: The identification of novel naphthyl and benzofuranyl amide analogs.. 26:2129-2132. 2016
Part 3: Notch-sparing -secretase inhibitors: SAR studies of 2-substituted aminopyridopyrimidinones.. 26:2138-2141. 2016
Discovery of adamantane based highly potent HDAC inhibitors.. 23:2532-2537. 2013
Novel diaryl ureas with efficacy in a mouse model of malaria.. 23:1022-1025. 2013
Anti-AIDS agents 87. New bio-isosteric dicamphanoyl-dihydropyranochromone (DCP) and dicamphanoyl-khellactone (DCK) analogues with potent anti-HIV activity.. 21:5831-5834. 2011
Organelle-selective energy transfer: a fluorescent indicator of intracellular environment.. 21:1849-1851. 2011
Design, synthesis and anticancer activity of piperazine hydroxamates and their histone deacetylase (HDAC) inhibitory activity.. 20:3906-3910. 2010
Genetic incorporation of an aliphatic keto-containing amino acid into proteins for their site-specific modifications.. 20:878-880. 2010
A retro-inverso TAT-like peptide designed to deliver cysteamine to cells.. 20:6321-6323. 2010
Functionalization of the 4,4-difluoro-4-bora-3a,4a-diaza-s-indacene (BODIPY) core.. 18:3112-3116. 2008
Structure-dependent inhibition of bladder and pancreatic cancer cell growth by 2-substituted glycyrrhetinic and ursolic acid derivatives.. 18:2633-2639. 2008
A diversity oriented synthesis of 3'-O-modified nucleoside triphosphates for DNA 'sequencing by synthesis'.. 16:3902-3905. 2006
Synthesis, biological activity, and X-ray crystal structural analysis of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 1: 4 '-substituted triclosan derivatives (vol 15, pg 5247, 2005). 16:3618-3619. 2006
Synthesis and biological activity of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 2: 2'-substituted triclosan derivatives.. 16:2163-2169. 2006
Synthesis of carbon-11 and fluorine-18 labeled N-acetyl-1-aryl-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline derivatives as new potential PET AMPA receptor ligands.. 16:2229-2233. 2006
Synthesis, biological activity, and X-ray crystal structural analysis of diaryl ether inhibitors of malarial enoyl acyl carrier protein reductase. Part 1: 4'-substituted triclosan derivatives.. 15:5247-5252. 2005
Synthesis and cytotoxic activity of 3-O-acyl/3-hydrazine /2-bromo/20,29-dibromo betulinic acid derivatives.. 14:4087-4091. 2004
Synthesis of 3-O-acyl/3-benzylidene/3-hydrazone/3-hydrazine/17-carboxyacryloyl ester derivatives of betulinic acid as anti-angiogenic agents.. 14:3169-3172. 2004
Betulinic acid and its derivatives as anti-angiogenic agents.. 14:2181-2184. 2004
Oligonucleotides with strongly fluorescent groups pi-conjugated to a nucleobase: syntheses, melting temperatures, and conformation.. 13:2785-2788. 2003
An efficient enzymatic synthesis of thiamin pyrophosphate.. 13:4139-4141. 2003
Stereochemical studies on phosphopantothenoylcysteine decarboxylase from Escherichia coli.. 13:339-342. 2003
The mechanism of action of bacimethrin, a naturally occurring thiamin antimetabolite.. 11:2245-2248. 2001
Dimeric beta-turn peptidomimetics as ligands for the neurotrophin receptor TrkC.. 11:207-210. 2001
Mechanistic studies on prolyl-4-hydroxylase: the vitamin C requiring uncoupled oxidation.. 10:1511-1514. 2000
Substrate and stereochemical specificity of the organophosphorus acid anhydrolase from Alteromonas sp. JD6.5 toward p-nitrophenyl phosphotriesters.. 10:1285-1288. 2000
Landomycin A inhibits DNA synthesis and G1/S cell cycle progression.. 9:1663-1666. 1999
Novel conformationally restricted tetracyclic analogs of delta8-tetrahydrocannabinol.. 9:2119-2124. 1999
A labeled guanidine ligand for studying sweet taste.. 8:881-884. 1998
Substrate specificity of human prolyl-4-hydroxylase.. 8:1139-1144. 1998
Acyclic nucleoside triphosphate analogs as terminators in biocatalytic DNA replication. 7:3013-3016. 1997
A small library of peptidomimetics to systematically vary and test the effects of X(1) constraints. 6:2761-2764. 1996
STEREOSPECIFIC ENZYMATIC-HYDROLYSIS OF PHOSPHORUS-SULFUR BONDS IN CHIRAL ORGANOPHOSPHATE TRIESTERS. 4:1473-1478. 1994
Structural basis for the differential RXR & RAR activity of stilbene retinoid analogs. 4:1447-1452. 1994
Synthesis and antiviral activity of a novel class of HIV-1 protease inhibitors containing a heterocyclic P1-P2 amide bond isostere. 4:2441-2446. 1994
Nonpeptide HIV protease inhibitors designed to replace a bound water. 3:2717-2722. 1993
Inactivation of HIV-1 protease by a tripeptidyl epoxide. 2:1441-1445. 1992
Phosphinic acid inhibitors of 3-hydroxy-3-methylglutaryl-coenzyme a reductase. 1:151-154. 1991
An efficient one-pot synthesis of tethered cyclohexadiene enaminonitriles from methyl-ketones: an effective route to quinazolines. 2008