Bioorganic and Medicinal Chemistry Journal

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An optimal "Click" formulation strategy for antibody-drug conjugate synthesis.. 28:115808-115808. 2020
In vitro and in silico elucidation of antidiabetic and anti-inflammatory activities of bioactive compounds from Momordica charantia L.. 27:3097-3109. 2019
Design and molecular modeling of novel P38 MAPK inhibitors targeting breast cancer, synthesized from oxygen heterocyclic natural compounds.. 27:1308-1319. 2019
Pyrrolizines: Design, synthesis, anticancer evaluation and investigation of the potential mechanism of action.. 25:5637-5651. 2017
A strategy for dual inhibition of the proteasome and fatty acid synthase with belactosin C-orlistat hybrids.. 25:2901-2916. 2017
Synthesis and molecular docking studies of new furochromone derivatives as p38 MAPK inhibitors targeting human breast cancer MCF-7 cells.. 25:2423-2436. 2017
Quinoxalinone (Part II). Discovery of (Z)-3-(2-(pyridin-4-yl)vinyl)quinoxalinone derivates as potent VEGFR-2 kinase inhibitors.. 24:1840-1852. 2016
Synthesis and evaluation of the 2,4-diaminoquinazoline series as anti-tubercular agents.. 22:6965-6979. 2014
Sulphonamide 1,4-dithia-7-azaspiro[4,4]nonane derivatives as gelatinase A inhibitors.. 21:7752-7762. 2013
DNA damage by C1027 involves hydrogen atom abstraction and addition to nucleobases.. 20:4744-4750. 2012
Design, synthesis, biological evaluation, and comparative Cox1 and Cox2 docking of p-substituted benzylidenamino phenyl esters of ibuprofenic and mefenamic acids.. 20:1259-1270. 2012
Probing DNA interstrand cross-link formation by an oxidized abasic site using nonnative nucleotides.. 19:5788-5793. 2011
The structure-activity relationship of urea derivatives as anti-tuberculosis agents.. 19:5585-5595. 2011
Anti-AIDS agents 84. Synthesis and anti-human immunodeficiency virus (HIV) activity of 2'-monomethyl-4-methyl- and 1'-thia-4-methyl-(3'R,4'R)-3',4'-di-O-(S)-camphanoyl-(+)-cis-khellactone (DCK) analogs.. 18:7203-7211. 2010
Discovery, synthesis, and biological evaluation of piperidinol analogs with anti-tuberculosis activity.. 17:3588-3594. 2009
Antitumor studies. Part 5: Synthesis, antitumor activity, and molecular docking study of 5-(monosubstituted amino)-2-deoxo-2-phenyl-5-deazaflavins.. 16:9161-9170. 2008
Antitumor studies. Part 4: Design, synthesis, antitumor activity, and molecular docking study of novel 2-substituted 2-deoxoflavin-5-oxides, 2-deoxoalloxazine-5-oxides, and their 5-deaza analogs.. 16:922-940. 2008
Novel triterpenoid from Citrus aurantium L. possesses chemopreventive properties against human colon cancer cells.. 16:5939-5951. 2008
Synthesis and cellular effects of cycloterpenals: cyclohexadienal-based activators of neurite outgrowth.. 16:7573-7581. 2008
Antitumor studies. part 3: design, synthesis, antitumor activity, and molecular docking study of novel 2-methylthio-, 2-amino-, and 2-(N-substituted amino)-10-alkyl-2-deoxo-5-deazaflavins.. 15:6336-6352. 2007
Radical scavenging and cytochrome P450 3A4 inhibitory activity of bergaptol and geranylcoumarin from grapefruit.. 15:3684-3691. 2007
Analgesic agents without gastric damage: Design and synthesis of structurally simple benzenesulfonanilide-type cyclooxygenase-1-selective inhibitors (vol 15, pg 1014, 2007). 15:3299-3300. 2007
Analgesic agents without gastric damage: design and synthesis of structurally simple benzenesulfonanilide-type cyclooxygenase-1-selective inhibitors.. 15:1014-1021. 2007
Inhibition of colon cancer cell growth and antioxidant activity of bioactive compounds from Poncirus trifoliata (L.) Raf.. 15:4923-4932. 2007
Antitumor studies. Part 1: design, synthesis, antitumor activity, and AutoDock study of 2-deoxo-2-phenyl-5-deazaflavins and 2-deoxo-2-phenylflavin-5-oxides as a new class of antitumor agents.. 15:242-256. 2007
Furocoumarins from grapefruit juice and their effect on human CYP 3A4 and CYP 1B1 isoenzymes.. 14:2606-2612. 2006
Stereoselective detoxification of chiral sarin and soman analogues by phosphotriesterase.. 9:2083-2091. 2001
Libraries of opiate and anti-opiate peptidomimetics containing 2,3-methanoleucine.. 5:1867-1871. 1997
Mapping the structural domains of E. coli carbamoyl phosphate synthetase using limited proteolysis.. 3:525-532. 1995