Rapid and efficient solid phase syntheses of cyclic peptides with endocyclic biaryl ether bonds Academic Article uri icon

abstract

  • Solid phase syntheses of the OF4949 derivatives 1 and 6 - 9 were performed via protection/deprotection of tyrosine side-chains on a support, and S(N)Ar macrocyclization reactions.

author list (cited authors)

  • Burgess, K., Lim, D., Bois-Choussy, M., & Zhu, J.

citation count

  • 41

publication date

  • May 1997